Melanotan 1jẹ afọwọṣe peptide sintetiki tiα-MSH (homonu ti o nmu alfa-melanocyte). O ṣiṣẹ nipasẹmu awọn olugba melanocortin-1 ṣiṣẹ (MC1R)lati lowoiṣelọpọ melanin, ẹbọ adayebapigmentation awọ araatiphotoprotection.
O ti jẹ bẹfọwọsi fun itọju erythropoietic protoporphyria (EPP)-aisan toje ti o fa ifamọ pupọ si imọlẹ oorun. Melanotan 1 ṣe iranlọwọ alekunifarada UV ina, dinkuphototoxic aati, ati ilọsiwajuaabo ara lodi si UV-induced bibajẹ.
YiyanMC1R agonist
Awọn ilọsiwajueumelanin iṣelọpọ
Peseadayeba oorun Idaabobo
Awọn atilẹyinAtunṣe DNA ati idahun egboogi-iredodo
O pọju funvitiligo, idena akàn ara, atiohun ikunra pigmentation
Ti ṣawari sinuegboogi-ti ogboatidermatological awọn itọju ailera
Mimo giga ≥99%
Iṣajọpọ peptide alakoso-lile (SPPS)
GMP-bi ẹrọ awọn ajohunše
Ipese iwọn: R&D si awọn ipele iṣowo