Orukọ | N- (n- glycylglyglyglyglycyl) Glycyl) -8-L-lysinvasopron |
Nọmba Com | 14636-12-5 |
Alolacular agbekalẹ | C52H74N16O15S2 |
Iwuwo Molucular | 1227.37 |
Nọmba Einecs | 238-680-8 |
Farabale | 1824.0 ± 65.0 ° C (asọtẹlẹ) |
Oriri | 1.46 ± 0.1 g / cm3 (asọtẹlẹ) |
Awọn ipo ipamọ | Jeki ni ibi dudu, afojusi inter, fipamọ ni firilser, labẹ -15 ° C. |
Onigbọwọ | (PKA) 9.90 ± 0.15 (asọtẹlẹ) |
[N--Triglycyl-8-Lereye] - 130: PN: WO2010033207se: 171Cheifedin. 1-triglycyl-8-lyseninivasopsosin; Nα-Glycyl-Glycyll- [8 -]]] laasisopour; Nα-Glycyl-Glycyl-lysinel-Lyssinsin; Nα-Glycyclyclyclycycylcylcylcylcylcyllcylcyly; Nα-Gly-Gly-Gly-8-lys-VosoPoPisin; Terlipopyin, terlipopini, terlipresse, Terlipressunam.
Terliperin, ti orukọ kemikali jẹ faspolylylylylylylylylylylylylysinsin, jẹ tuntun sintetiki ps sintetiki tuntun ti o n ṣiṣẹpọ tuntun-ṣiṣe ti o n ṣiṣẹda idaamu vasopin. O jẹ iru procug, eyiti ko ṣiṣẹ nipa ararẹ. O ṣe igbese nipasẹ Amipopeptitsese ni vivo si laiyara "Tu" tu "Vssing Lysopringjú Lẹhin yiyọ awọn iṣẹ ṣiṣe 3,000 mẹta ni N-Fertus. Nitorinaa, terliperess n ṣiṣẹ bi ifiomipamo ti o tu silẹ lasopromi ni oṣuwọn iduroṣinṣin.
Ipaniyan ipa ti terlipreti ni lati ṣe adehun finchnic iṣan iṣan ara ati dinku ṣiṣan ẹjẹ (bii idinku sisan ẹjẹ, ateri ti o dinku fun ṣiṣan ẹjẹ ti Ilu ati Iyipada Portal. Ni apa keji, o le dinku pilasima fun idojukọ reinma, nitorina o pọ si sisan ẹjẹ kikun, imudara iṣẹ kirin ati fifun urdrome irdrome. Terlipopire jẹ oogun nikan ti o le ṣe imudara oṣuwọn oṣuwọn iwalaaye ti awọn alaisan pẹlu prophogengeal varcesheageal varnorhage herorrrage. O ti lo ni akoko ti o lo ninu itọju ile-iwosan ti hemorrrage ti iyatọ. Ni afikun, Terlipreshin ti tun lo ni ifijišẹ ninu ẹdọ ati kidinrin. Ni gbogbogbo, o ṣee ṣe lati mu ipa ti o ni anfani ni mọnamọna iyalẹnu idaamu ati resuscitation carcitary. Ti a ṣe afiwe pẹlu Vasanres, o ni ipa ipa pipẹ, ko fa awọn ilolu ti o nira ati awọn ilolu to lagbara ninu eto inu ọkan ati ti o dara julọ fun itọju nla ati ibaramu fun itọju buburu ati ibaramu. Gba ati itọju ti awọn alaisan aisan ti o padanu.